GSK-J1
GSK-J1 is a highly potent H3K27 histone demethylase inhibitor with IC50 of 28 nM and 53 nM in cell-free assays for JMJD3 (KDM6B) and UTX (KDM6A), respectively, >10-fold selectivity over other tested demethylases.
| Catalog Number | T6847 |
| Alternative Name(s) | GSK J1 |
| Research Area | Chromatin/Epigenetic |
| Molecular Formula | C22H23N5O2 |
| CAS# | 1373422-53-7 |
| Purity | 99.67% |
| SMILES | OC(=O)CCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1 |
| Size | 25 mg |
| Supplier Page | https://www.targetmol.com/compound/GSK-J1 |
| Additional Information | https://www.targetmol.com/datasheet/T6847 |