Serabelisib (TAK-117)

Serabelisib (TAK-117, INK-1117, MLN-1117) is a potent and selective oral PI3Kα isoform inhibitor (IC50 of 21 nmol/L against PI3Kα) that has demonstrated > 100-fold selectivity relative to other class I PI3K family members (PI3Kβ/γ/δ) and mTOR, and a high degree of selectivity against many other kinase.

Price Not Available 5mg Serabelisib (TAK-117) Supplier Page

Trivial name	INK-1117, MLN-1117
Catalog Number	S8581
Molecular Formula	C19H17N5O3
CAS#	1268454-23-4
Inchi	InChI=1S/C19H17N5O3/c20-19-22-14-9-12(1-3-16(14)27-19)13-2-4-17-21-10-15(24(17)11-13)18(25)23-5-7-26-8-6-23/h1-4,9-11H,5-8H2,(H2,20,22)
Inchi Key	BLGWHBSBBJNKJO-UHFFFAOYSA-N
SMILES	C1COCCN1C(=O)C2=CN=C3N2C=C(C=C3)C4=CC5=C(C=C4)OC(=N5)N
Size	5mg
Supplier Page	http://www.selleckchem.com/products/tak-117-ink-1117-mln-1117.html
Additional Information	https://file.selleck.cn/downloads/struct/tak-117-ink-1117-mln-1117-chemical-structure-S8581.gif