Gilteritinib (ASP2215)

Gilteritinib (ASP2215) is a small-molecule FLT3/AXL inhibitor with IC50 values of 0.29 nM and 0.73 nM for FLT3 and AXL, respectively. It inhibits FLT3 at an IC50 value that was approximately 800-fold more potent than the concentration required to inhibit c-KIT (230 nM).

Price Not Available 100mg Gilteritinib (ASP2215) Supplier Page

Trivial name	N/A
Catalog Number	S7754
Molecular Formula	C29H44N8O3
CAS#	1254053-43-4
Inchi	InChI=1S/C29H44N8O3/c1-4-23-28(31-20-9-17-40-18-10-20)34-29(26(33-23)27(30)38)32-21-5-6-24(25(19-21)39-3)37-11-7-22(8-12-37)36-15-13-35(2)14-16-36/h5-6,19-20,22H,4,7-18H2,1-3H3,(H2,30,38)(H2,31,32,34)
Inchi Key	GYQYAJJFPNQOOW-UHFFFAOYSA-N
SMILES	CCC1=C(N=C(C(=N1)C(=O)N)NC2=CC(=C(C=C2)N3CCC(CC3)N4CCN(CC4)C)OC)NC5CCOCC5
Size	100mg
Supplier Page	http://www.selleckchem.com/products/gilteritinib-asp2215.html
Additional Information	https://file.selleck.cn/downloads/struct/gilteritinib-aps2215-chemical-structure-s7754.gif