Gandotinib (LY2784544)
Gandotinib (LY2784544) is a potent JAK2 inhibitor with IC50 of 3 nM, effective in JAK2V617F, 8- and 20-fold selective versus JAK1 and JAK3. Phase 2.
Trivial name | N/A |
Catalog Number | S2179 |
Molecular Formula | C13H15NO2S |
CAS# | 1229236-86-5 |
Inchi | InChI=1S/C13H15NO2S/c1-4-14-11-8-10(16-3)5-6-12(11)17-13(14)7-9(2)15/h5-8H,4H2,1-3H3/b13-7- |
Inchi Key | BGVLELSCIHASRV-QPEQYQDCSA-N |
SMILES | CCN1C2=C(C=CC(=C2)OC)SC1=CC(=O)C |
Size | 50mg |
Supplier Page | http://www.selleckchem.com/products/LY2784544.html |
Additional Information | https://file.selleck.cn/downloads/struct/LY2784544-chemical-structure-S2179.gif |