Gedatolisib (PKI-587)

Gedatolisib (PF-05212384, PKI-587) is a highly potent dual inhibitor of PI3Kα, PI3Kγ and mTOR with IC50 of 0.4 nM, 5.4 nM and 1.6 nM in cell-free assays, respectively. Phase 2.

Price Not Available 50mg Gedatolisib (PKI-587) Supplier Page

Trivial name	PF-05212384
Catalog Number	S2628
Molecular Formula	C28H28N4O3.HCl
CAS#	1197160-78-3
Inchi	InChI=1S/C28H28N4O3.ClH/c1-30(2)15-18-11-12-31-16-21(19-7-3-5-9-23(19)31)25-26(28(34)29-27(25)33)22-17-32(13-14-35-18)24-10-6-4-8-20(22)24;/h3-10,16-18H,11-15H2,1-2H3,(H,29,33,34);1H/t18-;/m0./s1
Inchi Key	NYQIEYDJYFVLPO-FERBBOLQSA-N
SMILES	CN(C)CC1CCN2C=C(C3=CC=CC=C32)C4=C(C5=CN(CCO1)C6=CC=CC=C65)C(=O)NC4=O.Cl
Size	50mg
Supplier Page	http://www.selleckchem.com/products/pki587.html
Additional Information	https://file.selleck.cn/downloads/struct/PKI-587-chemical-structure-s2628.gif