Aticaprant
Aticaprant (CERC-501, LY-2456302) is a potent, orally bioavailable, centrally-penetrant antagonist of the kappa opioid receptor with a Ki of 0.807 nM. It exhibits an antidepressant effect with the potential to treat major depressive disorder (MDD).
| Trivial name | CERC-501, LY-2456302 |
| Catalog Number | E4647 |
| Molecular Formula | C22H20ClN7O |
| CAS# | 1174130-61-0 |
| SMILES | C1CC(CNC1)N(C2=C(C=CC=N2)Cl)C(=O)C3=CC=C(C=C3)N4C5=C(C=CC=N5)N=N4 |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/aticaprant.html |
| Additional Information | https://file.selleck.cn/downloads/struct/E4647-Aticaprant-chemical-structure.png |