Aticaprant
Aticaprant (CERC-501, LY-2456302) is a potent, orally bioavailable, centrally-penetrant antagonist of the kappa opioid receptor with a Ki of 0.807 nM. It exhibits an antidepressant effect with the potential to treat major depressive disorder (MDD).
| Trivial name | CERC-501, LY-2456302 |
| Catalog Number | E4647 |
| Molecular Formula | C21H18BrNO3 |
| CAS# | 1174130-61-0 |
| SMILES | CC(=O)C1=CC2=C(C=C1)NC(C3C2C=CC3)C4=CC5=C(C=C4Br)OCO5 |
| Size | 1g |
| Supplier Page | http://www.selleckchem.com/products/aticaprant.html |
| Additional Information | https://file.selleck.cn/downloads/struct/E4647-Aticaprant-chemical-structure.png |