VU0238429

VU0238429 (M5 PAM) is the first positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5/M5) with EC50 of 1.16 μM at M5 and both > 30 μM at M1 and M3. VU0238429 shows no potentiator activity at M2 or M4.

Price Not Available 5mg VU0238429 Supplier Page

Trivial name	M5 PAM
Catalog Number	S2646
Molecular Formula	C24H29N5O3.C24H29NO5.5/2H2O.3Na
CAS#	1160247-92-6
SMILES	[Na+].[Na+].[Na+].CCCCC(=O)N(CC1=CC=C(C=C1)C2=CC=CC=C2C3=NN=N[NH]3)C(C(C)C)C(O)=O.CCOC(=O)C(C)CC(CC4=CC=C(C=C4)C5=CC=CC=C5)NC(=O)CCC(O)=O
Size	5mg
Supplier Page	http://www.selleckchem.com/products/vu0238429.html
Additional Information	https://file.selleck.cn/downloads/struct/vu0238429-chemical-structure-s2646.gif