Apabetalone (RVX-208)

Apabetalone (RVX-208, RVX-000222) is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2 in a cell-free assay, about 170-fold selectivity over BD1. Phase 2.

Price Not Available 10mM/1mL Apabetalone (RVX-208) Supplier Page

Trivial name	RVX-000222
Catalog Number	S7295
Molecular Formula	C20H22N2O5
CAS#	1044870-39-4
Inchi	InChI=1S/C20H22N2O5/c1-11-7-13(8-12(2)18(11)27-6-5-23)19-21-15-9-14(25-3)10-16(26-4)17(15)20(24)22-19/h7-10,23H,5-6H2,1-4H3,(H,21,22,24)
Inchi Key	NETXMUIMUZJUTB-UHFFFAOYSA-N
SMILES	CC1=CC(=CC(=C1OCCO)C)C2=NC3=C(C(=CC(=C3)OC)OC)C(=O)N2
Size	10mM/1mL
Supplier Page	http://www.selleckchem.com/products/rvx-208.html
Additional Information	https://file.selleck.cn/downloads/struct/RVX-208-chemical-structure-s7295.gif