MK-5046

MK-5046 is a potent, selective and orally active Bombesin receptor subtype-3 (BRS-3) allosteric agonist with an IC50 and an EC50 value of 27 and 25 nM for hBRS-3, respectively. MK-5046 inhibits food intake and reduces body weight of diet-induced obese (DIO) mouse models. MK-5046 can be used for the research of obesity.

Price Not Available 1mg MK-5046 Supplier Page
Catalog Number E7551
Molecular Formula C10H14N5O13P3.2Na
CAS# 1022152-70-0
Inchi InChI=1S/C10H16N5O13P3.2Na/c11-8-5-9(13-2-12-8)15(3-14-5)10-7(17)6(16)4(26-10)1-25-30(21,22)28-31(23,24)27-29(18,19)20;;/h2-4,6-7,10,16-17H,1H2,(H,21,22)(H,23,24)(H2,11,12,13)(H2,18,19,20);;/q;2*+1/p- 2/t4-,6-,7-,10-;;/m1../s1
Inchi Key TTWYZDPBDWHJOR-IDIVVRGQSA-L
SMILES C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)([O-])OP(=O)(O)[O-])O)O)N.[Na+].[Na+]
Size 1mg
Supplier Page http://www.selleckchem.com/products/mk-5046.html
Additional Information https://file.selleck.cn/downloads/struct/e7551-mk-5046-chemical-structure-tube.png