GSK0660
GSK0660 is a potent PPARβ/δ antagonist with a pIC50 of 6.8 (binding assay IC50 = 155 nM; antagonist assay IC50 = 300 nM) and is nearly inactive on PPARα and PPARγ with IC50s above approximately 10 μM.
| Trivial name | N/A |
| Catalog Number | S5817 |
| Molecular Formula | C19H18N2O5S2 |
| CAS# | 1014691-61-2 |
| Inchi | InChI=1S/C19H18N2O5S2/c1-25-16-12-14(20-13-6-4-3-5-7-13)8-9-15(16)21-28(23,24)17-10-11-27-18(17)19(22)26-2/h3-12,20-21H,1-2H3 |
| Inchi Key | NDFKBGWLUHKMFY-UHFFFAOYSA-N |
| SMILES | COC1=C(C=CC(=C1)NC2=CC=CC=C2)NS(=O)(=O)C3=C(SC=C3)C(=O)OC |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/gsk0660.html |
| Additional Information | https://file.selleck.cn/downloads/struct/gsk0660-chemical-structure-s5817.gif |