BMS-754807
BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.8 nM/1.7 nM in cell-free assays, less potent to Met (c-Met), Aurora A/B, TrkA/B and Ron, and shows little activity to Flt3, Lck, MK2, PKA, PKC etc. Phase 2.
| Trivial name | N/A |
| Catalog Number | S1124 |
| Molecular Formula | C27H40N8O7 |
| CAS# | 1001350-96-4 |
| Inchi | #N/A |
| Inchi Key | #N/A |
| SMILES | CC(C)C1N(C)C(=O)C(CC2=CC=CC=C2)NC(=O)C(CC(O)=O)NC(=O)CNC(=O)C(CCCNC(N)=N)NC1=O |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/BMS-754807.html |
| Additional Information | https://file.selleck.cn/downloads/struct/BMS-754807-chemical-structure-S1124.gif |
