Selleck Chemicals

Selleck Chemicals logo

Selleck Chemicals supplies over 3,000 inhibitors used in the study of cell signaling pathways. We actively tracks the latest science so our customers can rely on us to be the leading supplier of the newest inhibitors.

Company Website

Product Listing

8-Bromo-cAMP 25mg  | Purity Not Available

Selleck Chemicals

8-bromo-cAMP (8-Br-Camp) is a cell permeable analog of cAMP that activates cyclic-AMP-dependent protein kinase with a Ka value of 0.05 μM; and a PKA activator.

More Information Supplier Page

8-Bromo-cAMP 100mg  | Purity Not Available

Selleck Chemicals

8-bromo-cAMP (8-Br-Camp) is a cell permeable analog of cAMP that activates cyclic-AMP-dependent protein kinase with a Ka value of 0.05 μM; and a PKA activator.

More Information Supplier Page

8-Bromo-cAMP 10mM/1mL  | Purity Not Available

Selleck Chemicals

8-bromo-cAMP (8-Br-Camp) is a cell permeable analog of cAMP that activates cyclic-AMP-dependent protein kinase with a Ka value of 0.05 μM; and a PKA activator.

More Information Supplier Page

8-Bromo-cAMP 1g  | Purity Not Available

Selleck Chemicals

8-bromo-cAMP (8-Br-Camp) is a cell permeable analog of cAMP that activates cyclic-AMP-dependent protein kinase with a Ka value of 0.05 μM; and a PKA activator.

More Information Supplier Page

8-Cyclopentyl-1,3-dimethylxanthine 5mg  | Purity Not Available

Selleck Chemicals

8-Cyclopentyl-1,3-dimethylxanthine is a selective adenosine A1 receptor antagonist with Ki’s of 10.9 nM and 1440 nM for A1 receptor and A2 receptor, respectively.

More Information Supplier Page

8-Cyclopentyl-1,3-dimethylxanthine 25mg  | Purity Not Available

Selleck Chemicals

8-Cyclopentyl-1,3-dimethylxanthine is a selective adenosine A1 receptor antagonist with Ki’s of 10.9 nM and 1440 nM for A1 receptor and A2 receptor, respectively.

More Information Supplier Page

8-Gingerol 1mg  | Purity Not Available

Selleck Chemicals

8-Gingerol is a bioactive ingredient of ginger root (Zingiber officinale), a medicinal plant having anti-nausea, anti-inflammatory, and anti-carcinogenic properties and a carminative effect.

More Information Supplier Page

8-Hydroxyquinoline 100mg  | Purity Not Available

Selleck Chemicals

8-Hydroxyquinoline (8-Oxychinolin, 8-Quinolinol, Oxine) is an antiseptic with mild fungistatic, bacteriostatic, anthelmintic, and amebicidal action. It is also used as a reagent and metal chelator, as a carrier for radio-indium for diagnostic purposes.

More Information Supplier Page

8-Hydroxyquinoline 500mg  | Purity Not Available

Selleck Chemicals

8-Hydroxyquinoline (8-Oxychinolin, 8-Quinolinol, Oxine) is an antiseptic with mild fungistatic, bacteriostatic, anthelmintic, and amebicidal action. It is also used as a reagent and metal chelator, as a carrier for radio-indium for diagnostic purposes.

More Information Supplier Page

8-O-acetyl shanzhiside methyl ester 1mg  | Purity Not Available

Selleck Chemicals

8-O-acetyl shanzhiside methyl ester (Barlerin, ND01), isolated from the leaves of Lamiophlomis rotata Kudo, promotes angiogenesis, which leads to the improvement of functional outcome after stroke.8-O-Acetyl shanzhiside methyl ester can inhibts NF-κB.

More Information Supplier Page

8-OH-DPAT (8-Hydroxy-DPAT) 5mg  | Purity Not Available

Selleck Chemicals

8-OH-DPAT (8-Hydroxy-DPAT) is a kind of classic 5-HT1A agonist with the pIC50 of 8.19. It has a selectivity of almost-1000 fold for a subtype of the 5-HT1 binding site; Its biological half-life is 1.5 hous.

More Information Supplier Page

8-OH-DPAT (8-Hydroxy-DPAT) 100mg  | Purity Not Available

Selleck Chemicals

8-OH-DPAT (8-Hydroxy-DPAT) is a kind of classic 5-HT1A agonist with the pIC50 of 8.19. It has a selectivity of almost-1000 fold for a subtype of the 5-HT1 binding site; Its biological half-life is 1.5 hous.

More Information Supplier Page

8-OH-DPAT (8-Hydroxy-DPAT) 1g  | Purity Not Available

Selleck Chemicals

8-OH-DPAT (8-Hydroxy-DPAT) is a kind of classic 5-HT1A agonist with the pIC50 of 8.19. It has a selectivity of almost-1000 fold for a subtype of the 5-HT1 binding site; Its biological half-life is 1.5 hous.

More Information Supplier Page

9-amino-CPT (9-Aminocamptothecin) 5mg  | Purity Not Available

Selleck Chemicals

9-amino-CPT (9-Aminocamptothecin, 9-AC, Aminocamptothecin, 9-amino-20(S)-camptothecin) is a Topoisomerase I inhibitor with potent anticancer activities. 9-amino-CPT (9-Aminocamptothecin) is an active, water-insoluble derivative of camptothecin.

More Information Supplier Page

9-Aminoacridine 25mg  | Purity Not Available

Selleck Chemicals

9-Aminoacridine (Aminacrine) is a highly fluorescent dye used clinically as a topical antiseptic and experimentally as a mutagen, an intracellular pH indicator and a negative mode small molecule MALDI matrix.

More Information Supplier Page

9-Methoxycanthin-6-one 5mg  | Purity Not Available

Selleck Chemicals

9-Methoxycanthin-6-one is present in intact plant parts and in callus tissues of different explants with anti-tumour activity.

More Information Supplier Page

9-Phenanthrol 5mg  | Purity Not Available

Selleck Chemicals

9-Phenanthrol (9-Hydroxyphenanthrene, Phenanthren-9-o, 9-Phenanthrenol) is a selective TRPM4 inhibitor with an IC50 in the range of 0.02 μM, without effects on TRPM5.

More Information Supplier Page

9”-Methyl salvianolate B 5mg  | Purity Not Available

Selleck Chemicals

9”-Methyl salvianolate B (9′-methyllithospermate B, 9′-Methyl lithospermate B, 9”’-Methyl salvianolate B) is an active constituent in ethanol extract of Radix Salviae Miltiorrhizae.

More Information Supplier Page

9”-Methyl salvianolate B 1mg  | Purity Not Available

Selleck Chemicals

9”-Methyl salvianolate B (9′-methyllithospermate B, 9′-Methyl lithospermate B, 9”’-Methyl salvianolate B) is an active constituent in ethanol extract of Radix Salviae Miltiorrhizae.

More Information Supplier Page

A-1155463 5mg  | Purity Not Available

Selleck Chemicals

A-1155463 is a highly potent and selective BCL-XL inhibitor with EC50 of 65 nM in H146 cells.

More Information Supplier Page

A-1155463 25mg  | Purity Not Available

Selleck Chemicals

A-1155463 is a highly potent and selective BCL-XL inhibitor with EC50 of 65 nM in H146 cells.

More Information Supplier Page

A-1155463 Dihydrochloride 10mM/1mL  | Purity Not Available

Selleck Chemicals

A-1155463 Dihydrochloride, a highly potent and selective BCL-XL inhibitor, shows picomolar binding affinity to BCL-XL, and >1000-fold weaker binding to BCL-2 and related proteins BCL-W(Ki=19 nM) and MCL-1(Ki>440 nM).

More Information Supplier Page

A-1155463 Dihydrochloride 5mg  | Purity Not Available

Selleck Chemicals

A-1155463 Dihydrochloride, a highly potent and selective BCL-XL inhibitor, shows picomolar binding affinity to BCL-XL, and >1000-fold weaker binding to BCL-2 and related proteins BCL-W(Ki=19 nM) and MCL-1(Ki>440 nM).

More Information Supplier Page

A-1155463 Dihydrochloride 25mg  | Purity Not Available

Selleck Chemicals

A-1155463 Dihydrochloride, a highly potent and selective BCL-XL inhibitor, shows picomolar binding affinity to BCL-XL, and >1000-fold weaker binding to BCL-2 and related proteins BCL-W(Ki=19 nM) and MCL-1(Ki>440 nM).

More Information Supplier Page

A-1210477 100mg  | Purity Not Available

Selleck Chemicals

A-1210477 is a potent and selective MCL-1 inhibitor with Ki and IC50 of 0.454 nM and 26.2 nM, respectively, >100-fold selectivity over other Bcl-2 family members.

More Information Supplier Page

A-1210477 1g  | Purity Not Available

Selleck Chemicals

A-1210477 is a potent and selective MCL-1 inhibitor with Ki and IC50 of 0.454 nM and 26.2 nM, respectively, >100-fold selectivity over other Bcl-2 family members.

More Information Supplier Page

A-1210477 5mg  | Purity Not Available

Selleck Chemicals

A-1210477 is a potent and selective MCL-1 inhibitor with Ki and IC50 of 0.454 nM and 26.2 nM, respectively, >100-fold selectivity over other Bcl-2 family members.

More Information Supplier Page

A-1210477 25mg  | Purity Not Available

Selleck Chemicals

A-1210477 is a potent and selective MCL-1 inhibitor with Ki and IC50 of 0.454 nM and 26.2 nM, respectively, >100-fold selectivity over other Bcl-2 family members.

More Information Supplier Page

A-1331852 100mg  | Purity Not Available

Selleck Chemicals

A-1331852 is a potent and selectiveBCL-XL inhibitor with Ki value less than 0.01 nM for BCL-XL and 6 nM, 4 nM, 142 nM for Bcl-2, Bcl-W, MCL-1 respectively. It may be useful in the treatment of cancer, immune and autoimmune diseases.

More Information Supplier Page

A-1331852 1g  | Purity Not Available

Selleck Chemicals

A-1331852 is a potent and selectiveBCL-XL inhibitor with Ki value less than 0.01 nM for BCL-XL and 6 nM, 4 nM, 142 nM for Bcl-2, Bcl-W, MCL-1 respectively. It may be useful in the treatment of cancer, immune and autoimmune diseases.

More Information Supplier Page

A-1331852 10mM/1mL  | Purity Not Available

Selleck Chemicals

A-1331852 is a potent and selectiveBCL-XL inhibitor with Ki value less than 0.01 nM for BCL-XL and 6 nM, 4 nM, 142 nM for Bcl-2, Bcl-W, MCL-1 respectively. It may be useful in the treatment of cancer, immune and autoimmune diseases.

More Information Supplier Page

A-1331852 5mg  | Purity Not Available

Selleck Chemicals

A-1331852 is a potent and selectiveBCL-XL inhibitor with Ki value less than 0.01 nM for BCL-XL and 6 nM, 4 nM, 142 nM for Bcl-2, Bcl-W, MCL-1 respectively. It may be useful in the treatment of cancer, immune and autoimmune diseases.

More Information Supplier Page

A-1331852 25mg  | Purity Not Available

Selleck Chemicals

A-1331852 is a potent and selectiveBCL-XL inhibitor with Ki value less than 0.01 nM for BCL-XL and 6 nM, 4 nM, 142 nM for Bcl-2, Bcl-W, MCL-1 respectively. It may be useful in the treatment of cancer, immune and autoimmune diseases.

More Information Supplier Page

A-196 2mg  | Purity Not Available

Selleck Chemicals

A-196 is a potent and selective inhibitor of SUV420H1 and SUV420H2 with IC50 values of 0.025 and 0.144 μM, respectively; more than 100-fold selective over other histone methyltransferases and non-epigenetic targets.

More Information Supplier Page

A-196 5mg  | Purity Not Available

Selleck Chemicals

A-196 is a potent and selective inhibitor of SUV420H1 and SUV420H2 with IC50 values of 0.025 and 0.144 μM, respectively; more than 100-fold selective over other histone methyltransferases and non-epigenetic targets.

More Information Supplier Page

A-196 10mM/1mL  | Purity Not Available

Selleck Chemicals

A-196 is a potent and selective inhibitor of SUV420H1 and SUV420H2 with IC50 values of 0.025 and 0.144 μM, respectively; more than 100-fold selective over other histone methyltransferases and non-epigenetic targets.

More Information Supplier Page

A-205804 50mg  | Purity Not Available

Selleck Chemicals

A-205804 is a potent and selective inhibitor of E-selectin and ICAM-1 expression with IC50 of 20 nM and 25 nM respectively.

More Information Supplier Page

A-205804 10mg  | Purity Not Available

Selleck Chemicals

A-205804 is a potent and selective inhibitor of E-selectin and ICAM-1 expression with IC50 of 20 nM and 25 nM respectively.

More Information Supplier Page

A-3 hydrochloride 5mg  | Purity Not Available

Selleck Chemicals

A-3 hydrochloride, a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases, againsts cAMP-dependent protein kinase (PKA) (Ki=4.3 µM), casein kinase II (CK2) (Ki=5.1 µM) and myosin light chain kinase (MLCK) (Ki=7.4 µM), also inhibits Protein Kinase C (PKC) and casein kinase I (CK1) with Ki values of 47 µM and 80 µM, respectively.

More Information Supplier Page

A-317491 5mg  | Purity Not Available

Selleck Chemicals

A-317491 is a novel potent and selective non-nucleotide antagonist of P2X3 and P2X2/3 receptors with Ki values of 22 nM and 9 nM for human P2X3 and P2X2/3 receptors.

More Information Supplier Page

A-317491 25mg  | Purity Not Available

Selleck Chemicals

A-317491 is a novel potent and selective non-nucleotide antagonist of P2X3 and P2X2/3 receptors with Ki values of 22 nM and 9 nM for human P2X3 and P2X2/3 receptors.

More Information Supplier Page

A-366 10mM/1mL  | Purity Not Available

Selleck Chemicals

A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor with IC50 of 3.3nM and 38nM, exhibiting >1000-fold selectivity for G9a/GLP over 21 other methyltransferases.

More Information Supplier Page

A-366 10mg  | Purity Not Available

Selleck Chemicals

A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor with IC50 of 3.3nM and 38nM, exhibiting >1000-fold selectivity for G9a/GLP over 21 other methyltransferases.

More Information Supplier Page

A-366 50mg  | Purity Not Available

Selleck Chemicals

A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor with IC50 of 3.3nM and 38nM, exhibiting >1000-fold selectivity for G9a/GLP over 21 other methyltransferases.

More Information Supplier Page

A-443654 5mg  | Purity Not Available

Selleck Chemicals

A-443654, a derivative of indazole–pyridine compounds, is a pan Akt (Akt1, 2, & 3 isoforms) inhibitor which binds to the ATP-binding site of Akt. It is an ATP competitive and reversible inhibitor.

More Information Supplier Page