Telcagepant
Telcagepant (MK-0974) is an orally active calcitonin gene-related peptide (CGRP) receptor antagonist with Kis of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively.
| Trivial name | MK-0974 |
| Catalog Number | E7989 |
| Molecular Formula | C20H16ClN5O3 |
| CAS# | 781649-09-0 |
| Inchi | InChI=1S/C20H16ClN5O3/c1-22-19(27)16-10-12(6-8-23-16)11-29-20-17-15(7-9-28-17)18(25-26-20)24-14-4-2-13(21)3-5-14/h2-10H,11H2,1H3,(H,22,27)(H,24,25) |
| Inchi Key | QFCXANHHBCGMAS-UHFFFAOYSA-N |
| SMILES | CNC(=O)C1=NC=CC(=C1)COC2=NN=C(C3=C2OC=C3)NC4=CC=C(C=C4)Cl |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/telcagepant.html |
| Additional Information | https://file.selleck.cn/downloads/struct/e7989-telcagepant-chemical-structure-tube.png |