phentolamine hydrochloride

Phentolamine hydrochloride is a potent, selective, and orally active antagonist of α1 and α2 adrenergic receptors , with pKi values of 8.8, 8.0, and 8.3 for the human α2A, α2B, and α2C adrenergic receptors, respectively. It also shows binding affinities for the α1-adrenoceptor subtypes, exhibiting Ki values of 6.1 nM for cloned α1A/D, 39.8 nM for α1B, and 2.8 nM for α1C.

Price Not Available 25mg phentolamine hydrochloride Supplier Page

Catalog Number	E6046
Molecular Formula	C27H32N8O2
CAS#	73-05-2
Inchi	InChI=1S/C27H32N8O2/c1-5-13-34-25(36)21-18-28-26(29-19-9-11-20(12-10-19)33-16-14-32(4)15-17-33)31-24(21)35(34)23-8-6-7-22(30-23)27(2,3)37/h5-12,18,37H,1,13-17H2,2-4H3,(H,28,29,31)
Inchi Key	BKWJAKQVGHWELA-UHFFFAOYSA-N
SMILES	CC(C)(C1=NC(=CC=C1)N2C3=NC(=NC=C3C(=O)N2CC=C)NC4=CC=C(C=C4)N5CCN(CC5)C)O
Size	25mg
Supplier Page	http://www.selleckchem.com/products/phentolamine-hydrochloride.html
Additional Information	https://file.selleck.cn/downloads/struct/E6046-phentolamine-hydrochloride-chemical-structure.png