Mozavaptan (hydrochloride)

Mozavaptan hydrochloride(OPC 31260 HCl), a benzazepine derivative is a potent, selective, competitive, and orally active antagonist of vasopressin V2 receptor with an IC50 value of 14 nM. Mozavaptan hydrochloride shows ~85-fold selectivity for V2 receptor over V1 receptor. Mozavaptan hydrochloride has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone (SIADH), and congestive heart failure treatment.

Trivial name OPC 31260 HCl
Catalog Number E4957
Molecular Formula C13H16N2O2
CAS# 138470-70-9
Inchi InChI=1S/C13H16N2O2/c1-9(16)14-6-5-10-8-15-13-4-3-11(17-2)7-12(10)13/h3-4,7-8,15H,5-6H2,1-2H3,(H,14,16)
Inchi Key DRLFMBDRBRZALE-UHFFFAOYSA-N
SMILES CC(=O)NCCC1=CNC2=C1C=C(C=C2)OC
Size 5mg
Supplier Page http://www.selleckchem.com/products/mozavaptan-hydrochloride.html
Additional Information https://file.selleck.cn/downloads/struct/E4957-Mozavaptan-hydrochloride-chemical-structure.png