Cloperastine fendizoate
Cloperastine fendizoate (Hustazol) is a sedative used to relieve cough and also has a peripheral action that desensitizes the afferent nerves in the tracheobronchial region. It inhibits the hERG K+ currents in a concentration-dependent manner, with an IC50 value of 0.027 μM.
Trivial name | Hustazol |
Catalog Number | E4828 |
Molecular Formula | C26H23N5O |
CAS# | 85187-37-7 |
Inchi | InChI=1S/C26H23N5O/c1-26(32)14-19(15-26)25-30-22(23-24(27)28-11-12-31(23)25)18-8-7-17-9-10-20(29-21(17)13-18)16-5-3-2-4-6-16/h2-13,19,32H,14-15H2,1H3,(H2,27,28)/t19-,26+ |
Inchi Key | PKCDDUHJAFVJJB-VLZXCDOPSA-N |
SMILES | CC1(CC(C1)C2=NC(=C3N2C=CN=C3N)C4=CC5=C(C=C4)C=CC(=N5)C6=CC=CC=C6)O |
Size | 1g |
Supplier Page | http://www.selleckchem.com/products/cloperastine-fendizoate.html |
Additional Information | https://file.selleck.cn/downloads/struct/E4828-Cloperastine-fendizoate-chemical-structure.png |