PAR4 antagonist 2 | MedChemExpress (MCE)

PAR4 antagonist 2 (Compound 31) is a protease activated receptor 4 (PAR4) antagonist, with IC50 values of 95 nM and 367 nM for human PAR4 and mouse PAR4. PAR4 antagonist 2 is active against PAR4 activation by the native protease thrombin cleavage but not the synthetic PAR4 agonist peptide AYPGKF[1].

Trivial name PAR4 antagonist 2
Catalog Number HY-161401
Research Area Cardiovascular Disease
Purity ≥98.0%
SMILES O=C(NC1=NNC(C2=C(F)C=C(F)C=C2)=N1)C3=NN(C4=CC=CC=C4)C5=C3CCCC5
Size 1 mg
Supplier Page https://www.medchemexpress.com/par4-antagonist-2.html