PARP7/HDACs-IN-1 | MedChemExpress (MCE)

PARP7/HDACs-IN-1 (compound 9l) is a dual-target inhibitor targeting PARP7/HDAC with anti-tumor activity. PARP7/HDACs-IN-1 inhibits different subtypes of PARPs and HDACs with IC50s of 83.3 nM (PARP1), 3.1 nM (PARP7), 35 nM (HDAC1), 30.3 nM (HDAC2), 35.4 nM (HDAC3), and 6.4 nM respectively. (HDAC6)[1]. br/[1].

Trivial name PARP7/HDACs-IN-1
Catalog Number HY-162349
Research Area Cancer
Purity ≥98.0%
SMILES O=C1NN=CC(N[C@H](COCCC(N2CCN(CC2)C3=NC=C(C=N3)OCC4=CC=C(C=C4)/C=C/C(NO)=O)=O)C)=C1C(F)(F)F
Size 1 mg
Supplier Page https://www.medchemexpress.com/parp7-hdacs-in-1.html