PPARδ agonist 10 | MedChemExpress (MCE)

PPARδ agonist 10 (compound 7) is an orally active, selective, and partial agonist of PPARδ, with EC50 values of 0.053 μM and 0.30 µM for hPPARδ(LBD)-GAL4 and mPPARδ, respectively. PPARδ agonist 10 is a partial PPARδ agonist in transactivation assay but a full agonist on free fatty acids (FFA) oxidation in muscle cells both in vitro and in vivo. PPARδ agonist 10 can be used for dyslipidemia research[1].

Trivial name PPARδ agonist 10
Catalog Number HY-121542
Research Area Metabolic Disease
CAS# 685139-10-0
Purity ≥98.0%
SMILES O=C(COC1=CC=C(C=C1Cl)SC/C=C(C2=CC=C(C=C2)Br)/C3=CC=C(C=C3)Br)O
Size 1 mg
Supplier Page https://www.medchemexpress.com/pparδ-agonist-10.html