CI-988 hemihydrate | MedChemExpress (MCE)
CI-988 hemihydrate (PD134308) is a potent, selective and orally active CCK2R (cholecystokinin 2 receptor) antagonist with an IC50 of 1.7 nM for mouse cortex CCK2. CI-988 hemihydrate shows >1600-fold selectivity for CCK2 over CCK1 receptor. CI-988 hemihydrate has anxiolytic and anti-tumor effects[1][2][3].
| Trivial name | CI-988 hemihydrate |
| Catalog Number | HY-105226B |
| Alternative Name(s) | PD134308 hemihydrate |
| Research Area | Neurological Disease; Cancer |
| Purity | ≥98.0% |
| SMILES | OC(CCC(N[C@H](C1=CC=CC=C1)CNC([C@](CC2=CNC3=C2C=CC=C3)(C)NC(OC4[C@H]5C[C@H](C6)C[C@@H]4C[C@H]6C5)=O)=O)=O)=O.[1/2].O |
| Size | 1 mg |
| Supplier Page | https://www.medchemexpress.com/ci-988-hemihydrate.html |