Omarigliptin (MK-3102)

Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5).

Price Not Available 1g Omarigliptin (MK-3102) Supplier Page

Trivial name	N/A
Catalog Number	S8565
Molecular Formula	C17H20F2N4O3S
CAS#	1226781-44-7
Inchi	InChI=1S/C17H20F2N4O3S/c1-27(24,25)23-7-10-6-22(8-16(10)21-23)12-5-15(20)17(26-9-12)13-4-11(18)2-3-14(13)19/h2-4,7,12,15,17H,5-6,8-9,20H2,1H3/t12-,15+,17-/m1/s1
Inchi Key	MKMPWKUAHLTIBJ-ISTRZQFTSA-N
SMILES	CS(=O)(=O)N1C=C2CN(CC2=N1)C3CC(C(OC3)C4=C(C=CC(=C4)F)F)N
Size	1g
Supplier Page	http://www.selleckchem.com/products/omarigliptin-mk-3102.html
Additional Information	https://file.selleck.cn/downloads/struct/omarigliptin-mk-3102-chemical-structure-s8565.gif