umbralisib (TGR-1202)

Umbralisib (TGR-1202, Rp-5264), a novel, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 & 24.3 nM, respectively.

Price Not Available 100mg umbralisib (TGR-1202) Supplier Page

Trivial name	Rp-5264
Catalog Number	S8194
Molecular Formula	C31H24F3N5O3
CAS#	1532533-67-7
Inchi	InChI=1S/C31H24F3N5O3/c1-15(2)41-24-9-7-18(12-22(24)34)27-26-30(35)36-14-37-31(26)39(38-27)16(3)29-25(17-5-4-6-19(32)11-17)28(40)21-13-20(33)8-10-23(21)42-29/h4-16H,1-3H3,(H2,35,36,37)/t16-/m0/s1
Inchi Key	IUVCFHHAEHNCFT-INIZCTEOSA-N
SMILES	CC(C)OC1=C(C=C(C=C1)C2=NN(C3=NC=NC(=C23)N)C(C)C4=C(C(=O)C5=C(O4)C=CC(=C5)F)C6=CC(=CC=C6)F)F
Size	100mg
Supplier Page	http://www.selleckchem.com/products/tgr-1202.html
Additional Information	https://file.selleck.cn/downloads/struct/tgr-1202-chemical-structure-S8194.gif