GA-017

GA-017 inhibits theserine/threonine protein kinases large tumor suppressor kinase 1/2 (LATS1/2), which exerts inhibitory with IC50s against LATS1 and 2 of 4.10±0.79 and 3.92±0.42 nM, respectively, and competitively inhibits LATS1 and 2 against ATP, with Ki (inhibition constant) values of 0.58±0.11 and 0.25±0.03 nM, respectively.

Price Not Available 10mM/1mL GA-017 Supplier Page
Catalog Number E1145
Molecular Formula C18H21N3O4
CAS# 2351906-74-4
SMILES CC\C(=N\NC(=O)NCC1=CC(=CC=C1)O)C2=C(O)C(=C(O)C=C2)C
Size 10mM/1mL
Supplier Page http://www.selleckchem.com/products/ga-017.html
Additional Information https://file.selleck.cn/downloads/struct/e1145-ga-017-chemical-structure.gif