Relacorilant (CORT125134)
Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.
| Catalog Number | E1091 |
| Molecular Formula | C27H22F4N6O3S |
| CAS# | 1496510-51-0 |
| SMILES | C[N]1C=C(C=N1)[S;v6](=O)(=O)N2CCC3=CC4=C(CC3(C2)C(=O)C5=CC(=CC=N5)C(F)(F)F)C=N[N]4C6=CC=C(F)C=C6 |
| Size | 25mg |
| Supplier Page | http://www.selleckchem.com/products/relacorilant.html |
| Additional Information | https://file.selleck.cn/downloads/struct/e1091-relacorilant-chemical-structure.gif |