[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradykinin, CCK and bombesin receptors. Induces apoptosis and inhibits cancer cell growth in vitro.

Catalog Number | TP1931L1 |
Alternative Name(s) | [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base) |
Research Area | GPCR/G Protein |
Molecular Formula | C81H113N19O14 |
CAS# | TP1931L1 |
Purity | 97.68% |
SMILES | CC(C)C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=CC=C3)NC([C@@H](CC4=CNC5=C4C=CC=C5)NC([C@H](CCC(N)=O)NC([C@@H](CC6=CC=CC=C6)NC([C@H]7N(C([C@H](CCCCN)NC([C@H]8N(C([C@@H](CCCNC(N)=N)N)=O)CCC8)=O)=O)CCC7)=O)=O)=O)=O)=O)=O)=O.CC(O)=O |
Size | 1 mg |
Supplier Page | https://www.targetmol.com/compound/_D-Arg1,D-Phe5,D-Trp7,9,Leu11_-Substance P acetate |
Additional Information | https://www.targetmol.com/datasheet/TP1931L1 |