BI-3802
BI-3802 is a highly potent BCL6 degrader and inhibits the Bric-à-brac (BTB) domain of BCL6 with an IC50 value of ≤3 nM. BI-3802 induces the polymerization of BCL6 and promotes BCL6 degration depended on E3 ligase SIAH1. BI-3802 has antitumor activity[1][2].
| Catalog Number | T5408 |
| Research Area | Apoptosis |
| Molecular Formula | C24H29ClN6O3 |
| CAS# | 2166387-65-9 |
| SMILES | C[C@H](C[C@H](C)C1)CN1c(nc1)nc(Nc(cc2)cc(C=C3OCC(NC)=O)c2N(C)C3=O)c1Cl |
| Size | 5 mg |
| Supplier Page | https://www.targetmol.com/compound/BI_3802 |
| Additional Information | https://www.targetmol.com/datasheet/T5408 |
