CDK12-IN-E9
CDK12-IN-E9 is a potent and selective covalent CDK12 inhibitor and non-covalent CDK9 inhibitor while avoiding ABC transporter-mediated efflux. It has a weak binding ability to CDK7/CyclinH complex (IC50> 1 μM).

Catalog Number | T14915 |
Research Area | Cell Cycle/Checkpoint |
Molecular Formula | C24H30N6O2 |
CAS# | 2020052-55-3 |
SMILES | C(C)C1=C2N(C(NC3=CC(NC(C=C)=O)=CC=C3)=CC(=N2)N4[C@H](CCO)CCCC4)N=C1 |
Size | 1 mg |
Supplier Page | https://www.targetmol.com/compound/CDK12-IN-E9 |
Additional Information | https://www.targetmol.com/datasheet/T14915 |