CDK12-IN-E9

CDK12-IN-E9 is a potent and selective covalent CDK12 inhibitor and non-covalent CDK9 inhibitor while avoiding ABC transporter-mediated efflux. It has a weak binding ability to CDK7/CyclinH complex (IC50> 1 μM).

Price Not Available 1 mg CDK12-IN-E9 Supplier Page
Catalog Number T14915
Research Area Cell Cycle/Checkpoint
Molecular Formula C24H30N6O2
CAS# 2020052-55-3
SMILES C(C)C1=C2N(C(NC3=CC(NC(C=C)=O)=CC=C3)=CC(=N2)N4[C@H](CCO)CCCC4)N=C1
Size 1 mg
Supplier Page https://www.targetmol.com/compound/CDK12-IN-E9
Additional Information https://www.targetmol.com/datasheet/T14915