Birabresib (OTX015)
Birabresib (OTX015, MK 8628) is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4 in cell-free assays. Birabresib inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.
Trivial name | MK 8628 |
Catalog Number | S7360 |
CAS# | 202590-98-5 |
Size | 10mg |
Supplier Page | http://www.selleckchem.com/products/otx015.html |
Additional Information | https://file.selleck.cn/downloads/struct/OTX015-chemical-structure-s7360.gif |