Tazemetostat (EPZ-6438)
Tazemetostat (EPZ-6438, E7438) is a potent, and selective EZH2 inhibitor with Ki and IC50 of 2.5 nM and 11 nM in cell-free assays, exhibiting a 35-fold selectivity versus EZH1 and >4,500-fold selectivity relative to 14 other HMTs.
| Trivial name | E7438 |
| Catalog Number | S7128 |
| CAS# | 1403254-99-8 |
| Size | 10mg |
| Supplier Page | http://www.selleckchem.com/products/epz-6438.html |
| Additional Information | https://file.selleck.cn/downloads/struct/EPZ-6438-chemical-structure-s7128.gif |