RS-127445
RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.
| Trivial name | MT500 |
| Catalog Number | S2698 |
| Molecular Formula | C17H16FN3 |
| CAS# | 199864-87-4 |
| Inchi | InChI=1S/C17H16FN3/c1-10(2)15-9-16(21-17(19)20-15)13-7-8-14(18)12-6-4-3-5-11(12)13/h3-10H,1-2H3,(H2,19,20,21) |
| Inchi Key | ZZZQXCUPAJFVBN-UHFFFAOYSA-N |
| SMILES | CC(C)C1=NC(=NC(=C1)C2=CC=C(C3=CC=CC=C32)F)N |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/rs-127445.html |
| Additional Information | https://file.selleck.cn/downloads/struct/rs-127445-chemical-structure-s2698.gif |