PFI-1 (PF-6405761)

PFI-1 (PF-6405761) is a highly selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM and for BRD2 with IC50 of 98 nM in a cell-free assay.

Price Not Available 5mg PFI-1 (PF-6405761) Supplier Page
Trivial name N/A
Catalog Number S1216
Molecular Formula C19H20N4O3
CAS# 1403764-72-6
Inchi InChI=1S/C19H20N4O3/c1-20-19(24)11-22-18-10-21-14-6-4-12(8-15(14)23-18)13-5-7-16(25-2)17(9-13)26-3/h4-10H,11H2,1-3H3,(H,20,24)(H,22,23)
Inchi Key LYPCULYCGFOIDA-UHFFFAOYSA-N
SMILES CNC(=O)CNC1=CN=C2C=CC(=CC2=N1)C3=CC(=C(C=C3)OC)OC
Size 5mg
Supplier Page http://www.selleckchem.com/products/pfl-1.html
Additional Information https://file.selleck.cn/downloads/struct/PF-06405761-chemical-structure-s1216.gif