PFI-1 (PF-6405761)

PFI-1 (PF-6405761) is a highly selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM and for BRD2 with IC50 of 98 nM in a cell-free assay.

Price Not Available 5mg PFI-1 (PF-6405761) Supplier Page
Trivial name N/A
Catalog Number S1216
Molecular Formula C16H17N3O4S
CAS# 1403764-72-6
Inchi InChI=1S/C16H17N3O4S/c1-19-10-11-9-12(7-8-13(11)17-16(19)20)18-24(21,22)15-6-4-3-5-14(15)23-2/h3-9,18H,10H2,1-2H3,(H,17,20)
Inchi Key TXZPMHLMPKIUGK-UHFFFAOYSA-N
SMILES CN1CC2=C(C=CC(=C2)NS(=O)(=O)C3=CC=CC=C3OC)NC1=O
Size 5mg
Supplier Page http://www.selleckchem.com/products/pfl-1.html
Additional Information https://file.selleck.cn/downloads/struct/PF-06405761-chemical-structure-s1216.gif