Enarodustat (JTZ-951)
Enarodustat (JTZ-951) is a potent and orally active HIF prolyl hydroxylase inhibitor with IC50 of 0.22 μM for PHD2 and EC50 of 5.7 μM for EPO release from Hep3B cells. Enarodustat has the potential for the treatment of renal anemia.
| Trivial name | N/A |
| Catalog Number | S9656 |
| Molecular Formula | C17H16N4O4 |
| CAS# | 1262132-81-9 |
| SMILES | C1=CC=C(C=C1)CCC2=CC(=O)C(=C3N2NC=N3)C(=O)NCC(=O)O |
| Size | 25mg |
| Supplier Page | http://www.selleckchem.com/products/enarodustat.html |
| Additional Information | https://file.selleck.cn/downloads/struct/s9656-enarodustat-jtz-951--chemical-structure.gif |