Astemizole
Astemizole (R 43512) is a histamine H1-receptor antagonist with IC50 of 4.7 nM. Astemizole is also a potent inhibitor of ether à-go-go 1 (Eag1) and Eag-related gene (Erg) potassium channels. Astemizole has antineoplastic and antipruritic effects.
| Trivial name | R 43512 |
| Catalog Number | S0398 |
| Molecular Formula | C28H31FN4O |
| CAS# | 68844-77-9 |
| SMILES | COC1=CC=C(C=C1)CCN2CCC(CC2)NC3=NC4=CC=CC=C4N3CC5=CC=C(C=C5)F |
| Size | 25mg |
| Supplier Page | http://www.selleckchem.com/products/astemizole.html |
| Additional Information | https://file.selleck.cn/downloads/struct/s0398-astemizole-chemical-structure.gif |