Tropifexor (LJN452)
Tropifexor (LJN452) is a novel and highly potent agonist of FXR with EC50 of 0.2 nM in HTRF assay. It shows no significant off-target activity against a broad panel of enzyme, ion channel, nuclear receptor, and GPCR (>10000-fold selectivity for FXR).
| Trivial name | N/A |
| Catalog Number | S8733 |
| CAS# | 1383816-29-2 |
| Size | 2mg |
| Supplier Page | http://www.selleckchem.com/products/tropifexor-ljn452.html |
| Additional Information | https://file.selleck.cn/downloads/struct/tropifexor-ljn52-chemical-structure-s8733.gif |