CPI-360
CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
| Trivial name | N/A |
| Catalog Number | S7656 |
| Molecular Formula | C25H31N3O4 |
| CAS# | 1802175-06-9 |
| Inchi | InChI=1S/C25H31N3O4/c1-15-13-22(31-4)20(24(29)27-15)14-26-25(30)23-17(3)28(21-8-6-5-7-19(21)23)16(2)18-9-11-32-12-10-18/h5-8,13,16,18H,9-12,14H2,1-4H3,(H,26,30)(H,27,29)/t16-/m1/s1 |
| Inchi Key | PFPSFENQCNMITC-MRXNPFEDSA-N |
| SMILES | CC1=CC(=C(C(=O)N1)CNC(=O)C2=C(N(C3=CC=CC=C32)C(C)C4CCOCC4)C)OC |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/cpi-360.html |
| Additional Information | https://file.selleck.cn/downloads/struct/cpi-360-chemical-structure-s7656.gif |