GSK 5959
GSK5959 is a potent and selective BRPF1 bromodomain inhibitor with an IC50 of 80 nM and exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
| Trivial name | N/A |
| Catalog Number | S5916 |
| Molecular Formula | C51H63F2N11O10 |
| CAS# | 901245-65-6 |
| Inchi | #N/A |
| Inchi Key | #N/A |
| SMILES | CNC(=O)N1CCC2=C(C1)C(=N[N]2C3CCN(CC3)C(=O)CCOCCOCCOCCOCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)N7CCCC8=CC(=C(C=C78)C(F)F)C9=C[N](C)N=C9 |
| Size | 25mg |
| Supplier Page | http://www.selleckchem.com/products/gsk-5959.html |
| Additional Information | https://file.selleck.cn/downloads/struct/gsk-5959-chemical-structure-s5916.gif |