GSK 5959
GSK5959 is a potent and selective BRPF1 bromodomain inhibitor with an IC50 of 80 nM and exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
| Trivial name | N/A |
| Catalog Number | S5916 |
| Molecular Formula | C100H179N45O25 |
| CAS# | 901245-65-6 |
| Inchi | #N/A |
| Inchi Key | #N/A |
| SMILES | CC(C)CC(NC(=O)C(CC(O)=O)NC(=O)CNC(=O)CNC(=O)C(CCCNC(N)=N)NC(=O)C(CCCNC(N)=N)NC(=O)C(CCCNC(N)=N)NC(=O)C(CCC(N)=O)NC(=O)C(CCCNC(N)=N)NC(=O)C(CCCNC(N)=N)NC(=O)C(CCCCN)NC(=O)C(CCCCN)NC(=O)C(CCCNC(N)=N)NC(=O)CNNC(CC1=CC=C(O)C=C1)C=O)C(=O)NC(CC(C)C)C(=O)N2CCCC2C(=O)NC(CCCNC(N)=N)C(=O)NCC(=O)NC(CO)C(N)=O |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/gsk-5959.html |
| Additional Information | https://file.selleck.cn/downloads/struct/gsk-5959-chemical-structure-s5916.gif |