Sulfaphenazole
Sulfaphenazole (Depocid, Depotsulfonamide, Plisulfan, Raziosulfa) is an inhibitor of CYP2C9 with Ki value of 0.3 μM and demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki values of 63 and 29 μM for CYP2C8 and CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19).
| Trivial name | Depocid, Depotsulfonamide, Plisulfan, Raziosulfa |
| Catalog Number | S3673 |
| Molecular Formula | C24H24FN7O |
| CAS# | 526-08-9 |
| Inchi | InChI=1S/C24H24FN7O/c1-14(2)32-13-27-30-23(32)19-5-4-6-22(28-19)29-24(33)17-10-21(15(3)9-18(17)25)31-11-20(26-12-31)16-7-8-16/h4-6,9-14,16H,7-8H2,1-3H3,(H,28,29,33) |
| Inchi Key | YIDDLAAKOYYGJG-UHFFFAOYSA-N |
| SMILES | CC1=CC(=C(C=C1N2C=C(N=C2)C3CC3)C(=O)NC4=CC=CC(=N4)C5=NN=CN5C(C)C)F |
| Size | 25mg |
| Supplier Page | http://www.selleckchem.com/products/sulfaphenazole.html |
| Additional Information | https://file.selleck.cn/downloads/struct/sulfaphenazole-chemical-structure-s3673.gif |