Sulfaphenazole
Sulfaphenazole (Depocid, Depotsulfonamide, Plisulfan, Raziosulfa) is an inhibitor of CYP2C9 with Ki value of 0.3 μM and demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki values of 63 and 29 μM for CYP2C8 and CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19).
| Trivial name | Depocid, Depotsulfonamide, Plisulfan, Raziosulfa |
| Catalog Number | S3673 |
| Molecular Formula | C15H14N4O2S |
| CAS# | 526-08-9 |
| Inchi | InChI=1S/C15H14N4O2S/c16-12-6-8-14(9-7-12)22(20,21)18-15-10-11-17-19(15)13-4-2-1-3-5-13/h1-11,18H,16H2 |
| Inchi Key | QWCJHSGMANYXCW-UHFFFAOYSA-N |
| SMILES | C1=CC=C(C=C1)N2C(=CC=N2)NS(=O)(=O)C3=CC=C(C=C3)N |
| Size | 25mg |
| Supplier Page | http://www.selleckchem.com/products/sulfaphenazole.html |
| Additional Information | https://file.selleck.cn/downloads/struct/sulfaphenazole-chemical-structure-s3673.gif |