BX795
BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity is 140- and 1600-fold for PDK1 over PKA and PKC in cell-free assays, respectively. Meanwhile, the selectivity for PDK1 is 100-fold than GSK3β.
| Catalog Number | T1830 |
| Research Area | NF-Κb|||PI3K/Akt/mTOR signaling|||Tyrosine Kinase/Adaptors|||Cell Cycle/Checkpoint|||Autophagy |
| Molecular Formula | C23H26IN7O2S |
| CAS# | 702675-74-9 |
| SMILES | Ic1cnc(Nc2cc(NC(=O)N3CCCC3)ccc2)nc1NCCCNC(=O)c1cccs1 |
| Size | 10 mg |
| Supplier Page | https://www.targetmol.com/compound/BX795 |
| Additional Information | https://www.targetmol.com/datasheet/T1830 |