AM251
AM251 is a effective CB1 receptor antagonist (IC50/Ki: 8 /7.49 nM) that displays 306-fold selectivity over CB2 receptors; also effective GPR55 agonist (EC50: 39 nM).
| Catalog Number | T1915 |
| Research Area | GPCR/G Protein|||Endocrinology/Hormones |
| Molecular Formula | C22H21Cl2IN4O |
| CAS# | 183232-66-8 |
| Purity | 97.88% |
| SMILES | Cc1c(n(nc1C(=O)NN1CCCCC1)c1c(Cl)cc(Cl)cc1)c1ccc(I)cc1 |
| Size | 100 mg |
| Supplier Page | https://www.targetmol.com/compound/AM251 |
| Additional Information | https://www.targetmol.com/datasheet/T1915 |